SCHEMBL8554239

SCHEMBL8554239

COc1ccc2cc(C(C)CCC(O)CCc3cccnc3)ccc2c1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.48
CYP11B2 P19099 5/20 0.45
CYP11B1 P15538 4/20 0.45
PTAFR P25105 3/20 0.43
CYP19A1 P11511 2/20 0.43
CYP17A1 P05093 2/20 0.43
CYP2C9 P11712 1/20 0.43
GRM2 Q14416 2/20 0.43
IDO1 P14902 1/20 0.43
NAMPT P43490 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477516 0.86 CYP11B2 (0.51) CYP11B2CYP11B1PTAFRCYP19A1CYP17A1
SCHEMBL8484267 0.81 CYP11B2 (0.47) CYP11B2CYP11B1PTAFRCYP19A1CYP17A1
SCHEMBL8481502 0.76 CYP11B1 (0.40) CYP11B2CYP11B1PTAFRCYP19A1CYP17A1
SCHEMBL10695136 0.76 PTAFR (0.51) PTAFR
SCHEMBL5016747 0.74 CHRNA7 (0.57)
SCHEMBL10696517 0.73 KMT2A (0.49) CYP11B2CYP11B1PTAFRCYP19A1CYP2C9
SCHEMBL8479969 0.72 CYP51A1 (0.50) CYP11B2CYP11B1CYP19A1CYP17A1IDO1
SCHEMBL5752462 0.72 CYP11B2 (0.55) ABCB11CYP11B2CYP11B1CYP19A1CYP17A1
SCHEMBL8479757 0.72 POLB (0.52) NAMPTSMN1; SMN2
SCHEMBL8479585 0.72 CYP1A1 (0.59) ABCB11NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed