SCHEMBL8481502

SCHEMBL8481502

COCOc1ccc2cc(CCC(O)CCc3cccnc3)ccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.40
CYP11B2 P19099 4/20 0.40
CYP19A1 P11511 3/20 0.40
CYP2C9 P11712 1/20 0.40
NAMPT P43490 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
CYP51A1 Q16850 2/20 0.39
ALDH1A1 P00352 2/20 0.38
F9 P00740 1/20 0.38
F10 P00742 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
IDO1 P14902 1/20 0.38
PTAFR P25105 3/20 0.37
DHODH Q02127 1/20 0.37
CYP17A1 P05093 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477516 0.88 CYP11B2 (0.51) CYP11B1CYP11B2CYP19A1CYP2C9NAMPT
SCHEMBL8476422 0.84 LMNA (0.45) CYP11B1CYP11B2CYP19A1CYP2C9NAMPT
SCHEMBL8484267 0.83 CYP11B2 (0.47) CYP11B1CYP11B2CYP19A1CYP2C9HTR1A
SCHEMBL8481712 0.82 PTAFR (0.40) CYP11B1CYP11B2CYP19A1CYP2C9NAMPT
SCHEMBL8481721 0.82 PTAFR (0.40) CYP11B1CYP11B2CYP19A1CYP2C9NAMPT
SCHEMBL8479969 0.81 CYP51A1 (0.50) CYP11B1CYP11B2CYP19A1NAMPTMEN1
SCHEMBL8479757 0.79 POLB (0.52) NAMPTMEN1KMT2AALDH1A1POLB
SCHEMBL8073554 0.78 TBXAS1 (0.49) NAMPTMEN1KMT2AALDH1A1
SCHEMBL7954714 0.78 TBXAS1 (0.49) NAMPTMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL8482036 0.78 CYP19A1 (0.47) CYP11B1CYP11B2CYP19A1CYP51A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed