SCHEMBL8477516

SCHEMBL8477516

COc1ccc2cc(CCC(O)CCc3cccnc3)ccc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 7/20 0.51
CYP11B1 P15538 6/20 0.51
CYP19A1 P11511 2/20 0.51
CYP2C9 P11712 1/20 0.51
CYP17A1 P05093 2/20 0.49
IDO1 P14902 1/20 0.47
HTR1A P08908 1/20 0.46
DRD2 P14416 1/20 0.46
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
MAOA P21397 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8484267 0.94 CYP11B2 (0.47) CYP11B2CYP11B1CYP19A1CYP2C9CYP17A1
SCHEMBL8481502 0.88 CYP11B1 (0.40) CYP11B2CYP11B1CYP19A1CYP2C9CYP17A1
SCHEMBL8554239 0.86 ABCB11 (0.48) CYP11B2CYP11B1CYP19A1CYP2C9CYP17A1
SCHEMBL8479969 0.85 CYP51A1 (0.50) CYP11B2CYP11B1CYP19A1CYP17A1IDO1
SCHEMBL10695136 0.84 PTAFR (0.51) PTAFR
Hydrochloric Acid SCHEMBL8482036 0.82 CYP19A1 (0.47) CYP11B2CYP11B1CYP19A1CYP17A1IDO1
SCHEMBL10696517 0.81 KMT2A (0.49) CYP11B2CYP11B1CYP19A1CYP2C9RAB9A
SCHEMBL5016747 0.79 CHRNA7 (0.57) KDM4ECYP1A2
SCHEMBL8481869 0.78 KDM4E (0.53) CYP11B2CYP11B1CYP19A1CYP2C9IDO1
SCHEMBL7954714 0.78 TBXAS1 (0.49) SLC6A2SLC6A3NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed