SCHEMBL8554736

SCHEMBL8554736

O=C(c1ccc(F)cc1)C(F)Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
PTPN1 P18031 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
BCL2L1 Q07817 1/20 0.45
BAD Q92934 1/20 0.45
GSK3B P49841 3/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
LTA4H P09960 1/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
ALPG P10696 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364624 0.84 GSK3B (0.61) CES2CES1PTPN1CA1CA2
SCHEMBL28646814 0.82 CES2 (0.52) CES2CES1CA1CA2GSK3B
SCHEMBL18585299 0.81 CES2 (0.56) CES2CES1PTPN1CA1CA2
SCHEMBL31191256 0.81 CES2 (0.64) CES2CES1PTPN1CA1CA2
SCHEMBL28075917 0.80 CES2 (0.50) CES2CES1PTPN1CA1CA2
SCHEMBL27650390 0.80 CES2 (0.50) CES2CES1CA1CA2GSK3B
SCHEMBL1938267 0.80 CES2 (0.50) CES2CES1PTPN1CA1CA2
SCHEMBL27650405 0.80 ALDH1A1 (0.50) CES2CES1CA2GSK3BALDH1A1
SCHEMBL10580864 0.79 CES2 (0.54) CES2CES1PTPN1CA1CA2
SCHEMBL1110769 0.79 TDP1 (0.52) CES2CES1PTPN1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113880786-A Synthesis method and antioxidant application of camphene aldehyde thiazole hydrazone derivative 江西农业大学 2022-01-04 CN claimed
CN-115894461-B Novel coumarin-containing azole derivative, and preparation method and application thereof 沈阳药科大学 2024-01-23 CN disclosed
CN-116854683-A Coumarin thiazole derivative and preparation method and application thereof 中北大学 2023-10-10 CN disclosed
CN-115894461-A Novel coumarin azole-containing derivative and preparation method and application thereof 沈阳药科大学 2023-04-04 CN disclosed
CN-115745898-A Aromatic acrylamide-triazole compound, and preparation method and application thereof 许昌学院 2023-03-07 CN disclosed
CN-113880786-B Synthesis method and anti-oxidation application of camphene aldehyde thiazole hydrazone derivative 江西农业大学 2023-03-03 CN disclosed
CN-113880786-A Synthesis method and antioxidant application of camphene aldehyde thiazole hydrazone derivative 江西农业大学 2022-01-04 CN disclosed
CN-107625766-B Application of thiazole compound as antibacterial synergist 上海医药工业研究院 2021-08-31 CN disclosed
CN-103097367-A Phenylpropionic acid compound, preparation method therefor and medicinal use thereof INST PHARM & TOXICOLOGY AMMS 2013-05-08 CN disclosed
EP-0617031-B1 Orally active azole derivates URIACH & CIA SA J (ES) 1998-09-16 EP disclosed
WO-1998039330-A1 HETEROCYCLIC COMPOUNDS AS COX-2 INHIBITORS ABBOTT LABORATORIES (US) 1998-09-11 WO disclosed
US-5760245-A FUNGICIDES J. URIACH & CIA S.A. (ES) 1998-06-02 US disclosed
US-5646294-A FUNGICIDES J. URIACH & CIA. S.A. (ES) 1997-07-08 US disclosed
US-5478826-A Fungicides for human, animal and plants J. URIACH & CIA. S.A. (ES) 1995-12-26 US disclosed
EP-0617031-A1 Orally active azole derivates J. URIACH & CIA. S.A. (ES) 1994-09-28 EP disclosed
EP-0174769-B1 ANTIFUNGAL AZOLE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-11-21 EP disclosed
US-4925863-A 1,3-DI(1,2,4-TRIAZOL-1-YL)-2-PROPANOL DERIVATIVES SUBSTITUTED WITH A STYRYL GROUP IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-05-15 US disclosed
EP-0174769-A1 Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-03-19 EP disclosed