SCHEMBL8554805

SCHEMBL8554805

O=C(O)c1ccc(NC(=O)C(F)(F)F)nc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 17/20 0.59
HCAR2 Q8TDS4 2/20 0.49
P4HA1 P13674 1/20 0.47
P4HTM Q9NXG6 1/20 0.47
DEGS1 O15121 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21062101 0.87 HCAR3 (0.58) HCAR3HCAR2
SCHEMBL7094503 0.85 DEGS1 (0.46) HCAR3DEGS1L3MBTL1
SCHEMBL15065060 0.84 HCAR3 (0.54) HCAR3HCAR2P4HA1P4HTM
SCHEMBL10932719 0.81 HCAR3 (0.58) HCAR3HCAR2P4HA1P4HTM
SCHEMBL12903841 0.78 KDM4E (0.41) DEGS1L3MBTL1
SCHEMBL13656094 0.78 RAB9A (0.66) L3MBTL1
SCHEMBL6543272 0.78 ALDH1A1 (0.55) L3MBTL1
SCHEMBL2228695 0.78 PTGS1 (0.61) DEGS1L3MBTL1
SCHEMBL82675 0.77 HCAR3 (0.68) HCAR3HCAR2
SCHEMBL30753154 0.77 HCAR3 (0.65) HCAR3HCAR2P4HA1P4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed