SCHEMBL8555061

SCHEMBL8555061

O=C1[N]c2c(Br)cc(C(F)(F)F)cc2NC1=O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
JUN P05412 4/20 0.34
NFKB1 P19838 4/20 0.34
NFKB2 Q00653 4/20 0.34
RELA Q04206 4/20 0.34
ACE2 Q9BYF1 1/20 0.33
IKBKB O14920 1/20 0.31
GRM2 Q14416 1/20 0.30
GALR3 O60755 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6220507 0.84 GRM2 (0.31) IKBKBGRM2
SCHEMBL8130792 0.83 JUN (0.37) JUNNFKB1NFKB2RELAACE2
SCHEMBL3032750 0.81 JUN (0.39) JUNNFKB1NFKB2RELAACE2
SCHEMBL8557880 0.79 BCHE (0.31)
SCHEMBL8557193 0.78 HTR6 (0.35)
SCHEMBL8555364 0.75 HCAR1 (0.32)
SCHEMBL8556186 0.75
SCHEMBL8114995 0.73
SCHEMBL8124478 0.73
SCHEMBL9556590 0.71 JUN (0.43) JUNNFKB1NFKB2RELAACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP claimed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP claimed
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed