SCHEMBL8555243

SCHEMBL8555243

CC(O)CC(Oc1ccc(-c2ccccc2)cc1F)c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
ADRB3 P13945 3/20 0.40
ADRB1 P08588 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
NPY2R P49146 1/20 0.38
FAAH O00519 1/20 0.38
SLC6A4 P31645 3/20 0.37
ABCB1 P08183 2/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
KCNA5 P22460 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP17A1 P05093 2/20 0.36
SUCNR1 Q9BXA5 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555703 0.84 ADRB3 (0.47) ADRB3ADRB1FAAHMKNK1MKNK2
SCHEMBL8109544 0.83 SMN1; SMN2 (0.44) ADRB3ADRB1SMN1; SMN2SLC6A4KCNA5
SCHEMBL8550969 0.82 EPHX1 (0.46) ADRB3ADRB1SMN1; SMN2KCNA5
SCHEMBL8554047 0.81 SLC6A2 (0.51) SMN1; SMN2SLC6A4KCNA5CYP11B1CYP11B2
SCHEMBL8118264 0.80 DGAT2 (0.39) AKR1C3AKR1C2ADRB3ADRB1KCNA5
SCHEMBL8117056 0.79 CYP3A4 (0.40) AKR1C3AKR1C2ADRB3ADRB1KCNA5
SCHEMBL8552624 0.78 CYP19A1 (0.47) ADRB3ADRB1SMN1; SMN2MKNK1MKNK2
SCHEMBL8119038 0.77 CYP11B1 (0.43) ADRB3ADRB1CYP11B1CYP11B2
SCHEMBL8555652 0.77 PPARG (0.41) AKR1C3AKR1C2SMN1; SMN2KCNA5CYP11B1
SCHEMBL8552459 0.77 CYP17A1 (0.44) ADRB3ADRB1CYP11B1CYP11B2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed