SCHEMBL8555812

SCHEMBL8555812

O=C1[N]c2cc(I)ccc2NC1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 3/20 0.50
CES1 P23141 3/20 0.50
LRRK2 Q5S007 1/20 0.36
MAPT P10636 5/20 0.35
APP P05067 4/20 0.35
RAF1 P04049 3/20 0.35
MAP1LC3B Q9GZQ8 2/20 0.35
PLK4 O00444 2/20 0.35
EGFR P00533 1/20 0.35
NTRK1 P04629 1/20 0.35
ARAF P10398 1/20 0.35
PIM1 P11309 1/20 0.35
BRAF P15056 1/20 0.35
CSNK2A1 P68400 1/20 0.35
PIM3 Q86V86 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
MYOC Q99972 1/20 0.35
DYRK4 Q9NR20 1/20 0.35
SIRT3 Q9NTG7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4382993 0.81 TGM2 (0.44) TGM2CES1LRRK2MAPTAPP
SCHEMBL8556891 0.78 RET (0.37) TGM2CES1MAPTPIM1CSNK2A1
SCHEMBL8555842 0.78 KMT2A (0.39) TGM2CES1LRRK2MAPTMEN1
SCHEMBL5760370 0.78 ROS1 (0.46) TGM2CES1LRRK2MAPTMEN1
SCHEMBL2429783 0.75 JUN (0.44) NFKB1KMT2ATDP2PARP1
SCHEMBL8558339 0.75 PDPK1 (0.45) LRRK2EGFRCDK1KDRGSK3A
SCHEMBL8555149 0.74 CA1 (0.39) TGM2CES1HSD17B10TDP1PDE3B
SCHEMBL2334055 0.73 EPHX2 (0.41) TGM2CES1
SCHEMBL554552 0.72 MAPT (0.46) LRRK2MAPTPLK4PIM1MEN1
SCHEMBL8121209 0.70 GRIN2D (0.35) LRRK2MAPTPLK4MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed