SCHEMBL8558339

SCHEMBL8558339

N#Cc1ccc2c(c1)[N]C(=O)C(=O)N2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.45
CHEK1 O14757 1/20 0.38
PDGFRB P09619 8/20 0.38
KDR P35968 8/20 0.38
LRRK2 Q5S007 1/20 0.37
EGFR P00533 1/20 0.36
IMPDH2 P12268 1/20 0.36
IMPDH1 P20839 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
PGR P06401 1/20 0.35
GSK3B P49841 2/20 0.35
GSK3A P49840 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
NOTUM Q6P988 1/20 0.35
SNCA P37840 1/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555812 0.75 TGM2 (0.50) KDRLRRK2EGFRNOS1GSK3B
SCHEMBL5760370 0.75 ROS1 (0.46) PDPK1PDGFRBLRRK2CDK5CCNB2
SCHEMBL8556891 0.75 RET (0.37) PDPK1CHEK1
SCHEMBL8555842 0.75 KMT2A (0.39) LRRK2CCNB2CDK1CCNB1CCNB3
SCHEMBL2429783 0.72 JUN (0.44) NOTUM
SCHEMBL30639075 0.71 TGM2 (0.55) PDPK1LRRK2GSK3BGSK3ACDK5
SCHEMBL2498450 0.71 TGM2 (0.55) PDPK1LRRK2GSK3BGSK3ACDK5
SCHEMBL8555149 0.71 CA1 (0.39)
Hydrochloric Acid SCHEMBL11430847 0.70 TGM2 (0.53) PDPK1LRRK2GSK3BGSK3ACDK5
SCHEMBL2334055 0.70 EPHX2 (0.41) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed