SCHEMBL8556494

SCHEMBL8556494

N#CC1(N)CCc2ccc(Cl)cc2C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
PNMT P11086 1/20 0.38
SRD5A1 P18405 5/20 0.34
OTUD7B Q6GQQ9 1/20 0.34
BACE1 P56817 2/20 0.33
ESR1 P03372 4/20 0.33
ESR2 Q92731 4/20 0.33
OPRM1 P35372 1/20 0.33
SRD5A2 P31213 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16605572 0.82 BACE1 (0.42) KDM1APNMTBACE1
SCHEMBL8553587 0.78 BACE1 (0.39) KDM1ABACE1
Hydrochloric Acid SCHEMBL9179624 0.76 BACE1 (0.38) KDM1ABACE1
SCHEMBL16605583 0.75 KDM1A (0.41) KDM1APNMTBACE1ESR1ESR2
SCHEMBL8559759 0.72 KDM1A (0.41) KDM1AHTR2AHTR2CHTR2BPNMT
SCHEMBL8653266 0.70 ADRA2A (0.50) KDM1AHTR2AHTR2CPNMT
SCHEMBL27680709 0.67 KDM1A (0.43) KDM1AHTR2AHTR2CHTR2BSRD5A1
Hydrochloric Acid SCHEMBL9515919 0.67 KDM1A (0.40) KDM1AHTR2AHTR2CHTR2BPNMT
SCHEMBL2498788 0.66 ESR2 (0.51) KDM1AHTR2AHTR2CHTR2BSRD5A1
SCHEMBL15962624 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635497-B1 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR (FR) 1998-05-20 EP disclosed
US-5436261-A Adrenergic agonists ADIR ET COMPAGNIE (FR) 1995-07-25 US disclosed
EP-0635497-A2 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR ET COMPAGNIE (FR) 1995-01-25 EP disclosed