SCHEMBL8653266

SCHEMBL8653266

N#CC1(N)CCc2cccc(Cl)c2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.50
TAAR1 Q96RJ0 1/20 0.50
ADRA2B P18089 3/20 0.47
ADRA2C P18825 3/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
ADRA1B P35368 2/20 0.47
CYP2D6 P10635 1/20 0.39
PNMT P11086 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
KDM1A O60341 1/20 0.36
HTR1A P08908 2/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR7 P34969 2/20 0.32
HTR1B P28222 1/20 0.32
HTR6 P50406 1/20 0.32
HTR5A P47898 2/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
HTR1D P28221 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553587 0.76 BACE1 (0.39) ADRA2AKDM1A
Hydrochloric Acid SCHEMBL9179624 0.75 BACE1 (0.38) ADRA2AKDM1A
SCHEMBL7918142 0.73 BACE1 (0.33)
SCHEMBL8651098 0.73 ADRA2A (0.48) ADRA2ATAAR1ADRA2BADRA2CADRA1D
SCHEMBL8650675 0.73 LMNA (0.36)
SCHEMBL8648724 0.72 ADRA2A (0.47) ADRA2ATAAR1ADRA2BADRA2CADRA1D
SCHEMBL8649961 0.71 ADRA2A (0.46) ADRA2ATAAR1ADRA2BADRA2CADRA1D
SCHEMBL8828732 0.71 ADRA2A (0.46) ADRA2ATAAR1ADRA2BADRA2CADRA1D
SCHEMBL8556494 0.70 KDM1A (0.41) PNMTKDM1AHTR2AHTR2C
SCHEMBL8620656 0.70 ADRA2A (0.48) ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635495-B1 Benzospiroalkene derivates, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-09-16 EP disclosed
US-5648374-A A2-ADRENERGIC AGONISTS ADIR ET COMPAGNIE (FR) 1997-07-15 US disclosed
US-5486532-A ADRENERGIC AGONIST ADIR ET COMPAGNIE (FR) 1996-01-23 US disclosed
EP-0635495-A2 Benzospiroalkene derivates, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1995-01-25 EP disclosed