SCHEMBL8557090

SCHEMBL8557090

CN(c1ccc(F)cc1)S(=O)(=O)c1ccc2c(c1)CCC(C)(C)O2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.51
PKLR P30613 1/20 0.51
DAGLA Q9Y4D2 11/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 3/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
KCNH2 Q12809 2/20 0.47
ABHD6 Q9BV23 2/20 0.46
TRIM24 O15164 1/20 0.44
BRD1 O95696 1/20 0.44
BRPF1 P55201 1/20 0.44
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
FFAR1 O14842 1/20 0.43
NR1I2 O75469 1/20 0.42
DAGLB Q8NCG7 1/20 0.42
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557971 0.88 ATM (0.56) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL8558063 0.86 CYP3A4 (0.57) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL27481312 0.86 PKM (0.48) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL8557486 0.80 DAGLA (0.49) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL8553826 0.79 DAGLA (0.51) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL27482783 0.78 DAGLA (0.52) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL6025550 0.75 PKM (0.48) PKMPKLRKCNH2TRIM24BRD1
SCHEMBL4521621 0.74 PKM (0.58) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL3776603 0.74 PKM (0.58) PKMPKLRDAGLACYP3A4CYP2C19
SCHEMBL30511906 0.74 PKM (0.58) PKMPKLRDAGLACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1185153-A Benzopyrans and pharmaceutical composition contg. same CIBA GEIGY AG (CH) 1998-06-17 CN disclosed
EP-0828733-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Novartis AG (CH) 1998-03-18 EP disclosed
WO-1996037490-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NOVARTIS AG (CH) 1996-11-28 WO disclosed