SCHEMBL8557971

SCHEMBL8557971

CN(c1ccccc1)S(=O)(=O)c1ccc2c(c1)CCC(C)(C)O2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
DAGLA Q9Y4D2 11/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
KCNH2 Q12809 2/20 0.56
ABHD6 Q9BV23 2/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54
PKM P14618 2/20 0.50
PKLR P30613 1/20 0.50
NR1I2 O75469 1/20 0.47
DAGLB Q8NCG7 1/20 0.47
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
TRIM24 O15164 1/20 0.45
BRD1 O95696 1/20 0.45
BRPF1 P55201 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557090 0.88 PKM (0.51) ATML3MBTL1DAGLACYP3A4CYP2D6
SCHEMBL27481312 0.88 PKM (0.48) ATML3MBTL1DAGLACYP3A4CYP2D6
SCHEMBL8557486 0.87 DAGLA (0.49) ATML3MBTL1DAGLACYP3A4CYP2D6
SCHEMBL8558063 0.86 CYP3A4 (0.57) L3MBTL1DAGLACYP3A4CYP2D6CYP2C9
SCHEMBL8553826 0.86 DAGLA (0.51) ATML3MBTL1DAGLACYP3A4CYP2D6
SCHEMBL8487793 0.85 DAGLA (0.59) ATML3MBTL1DAGLACYP3A4CYP2D6
SCHEMBL8558762 0.85 DAGLA (0.56) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL27482783 0.82 DAGLA (0.52) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8557904 0.77 PKM (0.73) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL639690 0.76 PKM (0.58) DAGLACYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1185153-A Benzopyrans and pharmaceutical composition contg. same CIBA GEIGY AG (CH) 1998-06-17 CN disclosed
EP-0828733-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Novartis AG (CH) 1998-03-18 EP disclosed
WO-1996037490-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NOVARTIS AG (CH) 1996-11-28 WO disclosed