SCHEMBL8557486

SCHEMBL8557486

CN(c1cccnc1)S(=O)(=O)c1ccc2c(c1)CCC(C)(C)O2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 13/20 0.49
CYP2D6 P10635 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
KCNH2 Q12809 2/20 0.46
PKM P14618 2/20 0.45
PKLR P30613 1/20 0.45
ABHD6 Q9BV23 3/20 0.45
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NR1I2 O75469 1/20 0.42
DAGLB Q8NCG7 1/20 0.42
TRIM24 O15164 1/20 0.41
BRD1 O95696 1/20 0.41
BRPF1 P55201 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
MAPT P10636 1/20 0.39
PLCG2 P16885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27481312 0.87 PKM (0.48) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8557971 0.87 ATM (0.56) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8557090 0.80 PKM (0.51) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8553826 0.80 DAGLA (0.51) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8558063 0.78 CYP3A4 (0.57) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL7825817 0.75 HIF1A (0.49)
SCHEMBL8558762 0.75 DAGLA (0.56) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8487793 0.75 DAGLA (0.59) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL27482783 0.74 DAGLA (0.52) DAGLACYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL7820690 0.74 ATM (0.39) ATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1185153-A Benzopyrans and pharmaceutical composition contg. same CIBA GEIGY AG (CH) 1998-06-17 CN disclosed
EP-0828733-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Novartis AG (CH) 1998-03-18 EP disclosed
WO-1996037490-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NOVARTIS AG (CH) 1996-11-28 WO disclosed