SCHEMBL8557540

SCHEMBL8557540

COc1cccc(NCCCN)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.63
MTNR1B P49286 1/20 0.63
TAAR1 Q96RJ0 1/20 0.50
MAPT P10636 4/20 0.48
GAA P10253 1/20 0.48
ICMT O60725 3/20 0.48
RAB9A P51151 2/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
MAPK1 P28482 1/20 0.47
POLB P06746 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.47
NOS1 P29475 1/20 0.47
SYK P43405 1/20 0.46
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9148799 0.95 MTNR1A (0.61) MTNR1AMTNR1BTAAR1MAPTGAA
SCHEMBL15757422 0.91 MTNR1A (0.60) MTNR1AMTNR1BTAAR1MAPTICMT
SCHEMBL11114174 0.89 MTNR1A (0.66) MTNR1AMTNR1BMAPTGAAICMT
Propane SCHEMBL22639021 0.85 MTNR1A (0.57) MTNR1AMTNR1BMAPTICMTRAB9A
SCHEMBL11115757 0.84 MAPT (0.61) MTNR1AMTNR1BMAPTGAAICMT
SCHEMBL12520413 0.84 MTNR1B (0.60) MTNR1AMTNR1BMAPTICMTRAB9A
SCHEMBL10126890 0.84 MTNR1A (0.65) MTNR1AMTNR1BMAPTGAAICMT
SCHEMBL22631193 0.83 MAPT (0.54) MTNR1AMTNR1BMAPTMEN1KMT2A
SCHEMBL7505384 0.83 MTNR1B (0.59) MTNR1AMTNR1BMAPTICMTMEN1
SCHEMBL11117500 0.83 MTNR1A (0.59) MTNR1AMTNR1BMAPTICMTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1052723-C Bicyclic aromatic compounds as therapeutic agents KNOLL AG (DE) 2000-05-24 CN disclosed
EP-0876363-A1 POLYMER-BOUND FLUOROPHORES AS OPTICAL ION SENSORS Novartis AG (CH) 1998-11-11 EP disclosed
WO-1997011067-A1 POLYMER-BOUND FLUOROPHORES AS OPTICAL ION SENSORS NOVARTIS AG (CH) 1997-03-27 WO disclosed
CN-1133043-A Bicyclic aromatic compounds as therapeutic agents BOOTS CO PLC (DE) 1996-10-09 CN disclosed