SCHEMBL8557830

SCHEMBL8557830

COC(=O)C=Cc1nc2c(=O)[nH]c3ccccc3n2c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.43
POLB P06746 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
G6PD P11413 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
HKDC1 Q2TB90 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PDE4B Q07343 2/20 0.40
PDE2A O00408 1/20 0.40
PDE6D O43924 1/20 0.40
PDE8A O60658 1/20 0.40
PDE5A O76074 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555643 0.87 POLB (0.47) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8554710 0.80 POLB (0.50) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8557495 0.78 POLB (0.44) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8555929 0.78 POLB (0.46) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL9052411 0.74 POLB (0.55) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8553393 0.73 PDE2A (0.49) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8553821 0.73 POLB (0.49) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8557230 0.73 PDE5A (0.48) ADORA3MAPTPDE5APDE9A
SCHEMBL8034425 0.71 ADORA3 (0.61) ADORA3POLBKDM4EALDH1A1MAPT
SCHEMBL8554912 0.70 PDE5A (0.64) KDM4EALDH1A1MAPTNPSR1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed