SCHEMBL8557983

SCHEMBL8557983

Cc1ccc2c(c1)[nH]c(=O)c1nc(CO)c(C)n12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.43
ADORA3 P0DMS8 7/20 0.41
DDO Q99489 1/20 0.40
ADORA1 P30542 1/20 0.38
CHEK1 O14757 1/20 0.38
DAPK3 O43293 1/20 0.38
PRKD3 O94806 1/20 0.38
MET P08581 1/20 0.38
PDGFRA P16234 1/20 0.38
FLT1 P17948 1/20 0.38
LTK P29376 1/20 0.38
GRK5 P34947 1/20 0.38
CDK8 P49336 1/20 0.38
PRKX P51817 1/20 0.38
NEK2 P51955 1/20 0.38
LIMK1 P53667 1/20 0.38
CDK5 Q00535 1/20 0.38
ACVR1 Q04771 1/20 0.38
TYRO3 Q06418 1/20 0.38
PRKAA1 Q13131 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558719 0.88 ADORA3 (0.50) DAOADORA3ADORA1
SCHEMBL8557784 0.84 PDE5A (0.47) ALDH1A1TSHRCYP1A2CYP3A4CYP2C19
SCHEMBL8553393 0.84 PDE2A (0.49) ADORA3ADORA1ALDH1A1KDM4EHPGD
SCHEMBL4978084 0.72 ADORA3 (0.49) DAOADORA3DDOADORA1CHEK1
SCHEMBL8554724 0.71 PDE5A (0.48) CHEK1DAPK3PRKD3METPDGFRA
SCHEMBL8554829 0.71 PDE9A (0.61) TSHRCYP1A2CYP3A4CYP2C19KCNMA1
SCHEMBL8557272 0.70 CHEK1 (0.44) ADORA3CHEK1DAPK3PRKD3MET
SCHEMBL7506152 0.70 DAO (0.42) DAOADORA3DDOCHEK1DAPK3
SCHEMBL8556228 0.70 ADORA3 (0.50) ADORA3CHEK1DAPK3PRKD3MET
SCHEMBL7506016 0.69 CHEK1 (0.58) ADORA3CHEK1DAPK3PRKD3MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed