SCHEMBL8558001

SCHEMBL8558001

NS(=O)(=O)c1ccc(-c2cc(CCC(C(=O)O)c3ncco3)ccc2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSA P10619 7/20 0.41
PTGS2 P35354 6/20 0.38
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
CA4 P22748 1/20 0.37
PTGS1 P23219 5/20 0.36
GABRA2 P47869 2/20 0.35
CA5A P35218 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
MME P08473 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559917 0.91 CTSA (0.42) CTSAPTGS2GABRA2
SCHEMBL5733045 0.82 DRD1 (0.40) CTSAPTGS2CA1CA2CA12
SCHEMBL5732083 0.76 KMT2A (0.41) CTSAPTGS2CA1CA2CA12
SCHEMBL5732775 0.73 PTGS2 (0.42) CTSAPTGS2PTGS1
SCHEMBL8559048 0.72 PTGS2 (0.43) CTSAPTGS2PTGS1
SCHEMBL6002014 0.71 CA12 (0.48) CTSAPTGS2CA1CA2CA12
SCHEMBL5733199 0.70 CA2 (0.41) CA1CA2CA12CA9CA4
SCHEMBL6002042 0.70 CA1 (0.44) CTSAPTGS2CA1CA2CA12
SCHEMBL5734311 0.68 CA1 (0.49) PTGS2CA1CA2CA12CA9
SCHEMBL5733048 0.68 CA2 (0.41) CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719163-A ARTHRITIS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed