SCHEMBL8558181

SCHEMBL8558181

CCOC(=O)CCN1CCN(c2ccc(O)cc2)C1=O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.50
DRD2 P14416 5/20 0.46
DRD3 P35462 5/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
RAB9A P51151 1/20 0.44
HDAC1 Q13547 4/20 0.41
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
CYP1A1 P04798 2/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417017 0.88 DRD2 (0.52) S1PR1DRD2DRD3KDM4EGAA
SCHEMBL177341 0.83 S1PR1 (0.76) S1PR1DRD2DRD3HDAC1CYP1A1
SCHEMBL8561767 0.81 S1PR1 (0.45) S1PR1DRD2DRD3KMT2AMEN1
SCHEMBL8564103 0.80 S1PR1 (0.42) S1PR1DRD2DRD3LMNAKMT2A
SCHEMBL1410264 0.78 DRD2 (0.45) S1PR1DRD2DRD3LMNAHDAC1
SCHEMBL7281200 0.78 S1PR1 (0.44) S1PR1DRD2DRD3KMT2AMEN1
SCHEMBL31662444 0.77 RAB9A (0.47) S1PR1DRD2DRD3KMT2AMEN1
SCHEMBL31662551 0.77 DRD2 (0.48) S1PR1DRD2DRD3RAB9AHDAC1
SCHEMBL7284261 0.76 HRH2 (0.44) S1PR1DRD2DRD3KDM4ELMNA
SCHEMBL3712107 0.76 S1PR1 (0.48) S1PR1DRD2DRD3KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1048490-C Cyclic derivatives, pharmaceutical compositions containing these compounds and processes for preparing them THOMAE GMBH DR K (DE) 2000-01-19 CN disclosed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed