SCHEMBL8558200

SCHEMBL8558200

NC(N)=NS(=O)(=O)c1ccc(Cl)nc1Cl

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F2 P00734 20/20 0.49
PRSS1 P07477 20/20 0.49
PRSS2 P07478 20/20 0.49
PRSS3 P35030 20/20 0.49
LMNA P02545 1/20 0.42
AGO2 Q9UKV8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31028763 0.75 CA2 (0.37) LMNA
Hydrochloric Acid SCHEMBL28170640 0.73 NFE2L2 (0.34)
SCHEMBL11760774 0.73 NFE2L2 (0.34)
SCHEMBL11760766 0.73 NFE2L2 (0.34)
SCHEMBL30752415 0.72 TRPV4 (0.37)
SCHEMBL17368 0.72 TRPV4 (0.37)
SCHEMBL8558197 0.71 ALDH1A1 (0.31)
SCHEMBL22029021 0.71 NFE2L2 (0.38) LMNA
SCHEMBL30826830 0.71 NFE2L2 (0.38) LMNA
SCHEMBL10515229 0.70 F2 (0.59) F2PRSS1PRSS2PRSS3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed