SCHEMBL8558495

SCHEMBL8558495

Cc1cccc(S(=O)(=O)c2ccc(C(=N)N)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.46
ABCC8 Q09428 1/20 0.46
KCNJ11 Q14654 1/20 0.46
KCNJ8 Q15842 1/20 0.46
C1S P09871 1/20 0.45
F2 P00734 1/20 0.45
PRSS1 P07477 1/20 0.45
PRSS2 P07478 1/20 0.45
PRSS3 P35030 1/20 0.45
TMPRSS6 Q8IU80 2/20 0.44
MRGPRX1 Q96LB2 2/20 0.44
HTT P42858 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 1/20 0.43
NAMPT P43490 2/20 0.43
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558497 0.83 GAA (0.61) F2PRSS1PRSS2PRSS3TMPRSS6
SCHEMBL9029174 0.82 ALDH1A1 (0.45) F2MRGPRX1ALDH1A1MAPTHPGD
SCHEMBL8163851 0.80 CYP11B1 (0.43) C1SF2HTTALDH1A1MAPT
SCHEMBL8558127 0.80 F10 (0.47) F2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL9031533 0.80 F2 (0.51) F2PRSS1PRSS2PRSS3MRGPRX1
SCHEMBL31038387 0.79 GAA (0.67) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL6151129 0.79 GAA (0.67) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL822302 0.79 KMT2A (0.59) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL29468572 0.79 KMT2A (0.59) ABCC9ABCC8KCNJ11KCNJ8HTT
SCHEMBL8624231 0.79 C1S (0.41) ABCC9ABCC8KCNJ11KCNJ8C1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed