SCHEMBL8557792

SCHEMBL8557792

O=C(O)Oc1nc2c(=O)[nH]c3cc(C(F)(F)F)ccc3n2c1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.47
PDE9A O76083 2/20 0.47
NPBWR1 P48145 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
DGAT1 O75907 1/20 0.38
KCNH2 Q12809 1/20 0.38
TNKS O95271 2/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
MAPT P10636 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
HSP90AA1 P07900 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557199 0.88 PDE5A (0.43) PDE5APDE9AKDM4EALDH1A1HPGD
SCHEMBL8557418 0.85 PDE5A (0.49) PDE5APDE9AMEN1KMT2AMAPT
SCHEMBL8555764 0.85 PDE5A (0.49) PDE5APDE9ANPBWR1MEN1KMT2A
SCHEMBL8557015 0.82 PDE9A (0.47) PDE5APDE9AMEN1KMT2AMAPT
SCHEMBL8553493 0.80 PDE9A (0.58) PDE5APDE9ANPBWR1MEN1KMT2A
SCHEMBL8554950 0.80 PDE5A (0.44) PDE5APDE9AKDM4EALDH1A1HPGD
SCHEMBL8558570 0.77 KDM4E (0.48) PDE5APDE9AKMT2AMAPTCYP1A2
SCHEMBL8558977 0.75 PDE5A (0.38) PDE5APDE9AMGLL
SCHEMBL8557499 0.74 PDE5A (0.46) PDE5APDE9AMEN1KMT2ATNKS
SCHEMBL8553369 0.73 PDE5A (0.45) PDE5APDE9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP claimed
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed