SCHEMBL8559546

SCHEMBL8559546

O=C(Nc1cc(Cl)ccc1Cl)c1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.55
AVPR1A P37288 3/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
ACHE P22303 2/20 0.45
HSD17B3 P37058 1/20 0.45
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ALDH1A1 P00352 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
EPHX1 P07099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561645 0.92 AVPR2 (0.58) AVPR2AVPR1AACHENPSR1
SCHEMBL8557607 0.89 NPC1 (0.50) AVPR2AVPR1AALDH1A1NPSR1
SCHEMBL8561097 0.87 AVPR2 (0.52) AVPR2AVPR1AMEN1KMT2AHDAC1
SCHEMBL8563565 0.87 NAMPT (0.50) AVPR2AVPR1AMEN1KMT2AHDAC1
SCHEMBL8557503 0.84 ACHE (0.58) AVPR2AVPR1AACHEHSD17B3
SCHEMBL8558027 0.83 AVPR2 (0.69) AVPR2AVPR1A
SCHEMBL8563019 0.82 AVPR2 (0.59) AVPR2AVPR1AACHE
SCHEMBL8563344 0.81 AVPR2 (0.81) AVPR2AVPR1A
SCHEMBL8559349 0.81 AVPR2 (0.60) AVPR2AVPR1AACHE
SCHEMBL8562633 0.80 AVPR2 (0.55) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed