SCHEMBL8563565

SCHEMBL8563565

COc1ccc(Cl)c(NC(=O)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
RAB9A P51151 3/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 3/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
NPC1 O15118 2/20 0.45
KMT2A Q03164 2/20 0.45
AVPR2 P30518 1/20 0.45
AVPR1A P37288 1/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
F10 P00742 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556252 0.87 NAMPT (0.63) NAMPTSMN1; SMN2RAB9AKDM4EMAPT
SCHEMBL8559546 0.87 AVPR2 (0.55) HDAC1HDAC8HDAC6ALDH1A1KMT2A
SCHEMBL8557607 0.85 NPC1 (0.50) RAB9AMAPTALDH1A1NPC1AVPR2
SCHEMBL8561097 0.83 AVPR2 (0.52) NAMPTHDAC1HDAC8HDAC6SMN1; SMN2
SCHEMBL8558857 0.82 HPGD (0.57) NAMPTSMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8561645 0.81 AVPR2 (0.58) RAB9AKDM4ENPC1AVPR2AVPR1A
SCHEMBL8558377 0.81 NAMPT (0.54) NAMPTSMN1; SMN2RAB9AKDM4EMAPT
SCHEMBL8562633 0.78 AVPR2 (0.55) SMN1; SMN2RAB9ANPC1AVPR2AVPR1A
SCHEMBL8563019 0.78 AVPR2 (0.59) NAMPTAVPR2AVPR1A
SCHEMBL8562828 0.77 AVPR2 (0.49) SMN1; SMN2RAB9AMAPTNPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed