SCHEMBL8559747

SCHEMBL8559747

CCCn1ccc(NC(=O)C(NC(=O)OC(C)(C)C)c2ccc3c(c2)C(C)(C)CCC3(C)C)c1C(=O)OC

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.35
CYP26A1 O43174 4/20 0.35
RARB P10826 3/20 0.35
RARG P13631 3/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
RARA P10276 2/20 0.33
CYP26B1 Q9NR63 1/20 0.33
BACE1 P56817 4/20 0.32
AAK1 Q2M2I8 3/20 0.32
RXRA P19793 2/20 0.32
RXRB P28702 1/20 0.32
PPARG P37231 1/20 0.30
CTSL P07711 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102598 0.84 CTSS (0.34) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8106311 0.80 RARB (0.37) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8108607 0.77 RARB (0.35) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8108628 0.75 RARB (0.36) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8106743 0.74 MEN1 (0.42) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8558167 0.74 CTSS (0.40) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8757257 0.73 RARB (0.40) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8748829 0.72 RARB (0.55) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8100983 0.72 RARB (0.44) CYP3A4CYP26A1RARBRARGCTSS
SCHEMBL8748606 0.72 RARB (0.40) CYP3A4CYP26A1RARBRARGCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5709867-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, AND OPHTHALMOLOGICAL DISORDERS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1998-01-20 US disclosed