SCHEMBL8719948

SCHEMBL8719948

CCOC(=O)CC1CCN(C(=O)c2ccc(-c3ccc(C#N)cc3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 6/20 0.49
SLC6A7 Q99884 1/20 0.47
SIGMAR1 Q99720 1/20 0.46
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
EPHX2 P34913 1/20 0.46
ALDH1A1 P00352 1/20 0.45
CCNK O75909 1/20 0.45
CDK12 Q9NYV4 1/20 0.45
USP14 P54578 1/20 0.45
GAA P10253 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
PTGER4 P35408 1/20 0.43
PTGER2 P43116 1/20 0.43
PTGDR Q13258 1/20 0.43
FASN P49327 1/20 0.43
PDK1 Q15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8407569 0.89 CCNK (0.51) KDM1ASLC6A7SIGMAR1EPHX2ALDH1A1
SCHEMBL8410939 0.87 GRM3 (0.50) KDM1AHRH2HRH1HRH3ALDH1A1
SCHEMBL8568607 0.84 SLC6A7 (0.49) KDM1ASLC6A7SIGMAR1EPHX2ALDH1A1
SCHEMBL8410357 0.83 ITGB3 (0.51)
SCHEMBL8560134 0.82 KDM1A (0.49) KDM1AEPHX2ALDH1A1CCNKCDK12
SCHEMBL12156641 0.81 MGLL (0.48) GAA
SCHEMBL8544211 0.81 ACHE (0.56) ALDH1A1GAA
SCHEMBL8430024 0.81 ALDH1A1 (0.56) KDM1ASLC6A7SIGMAR1EPHX2ALDH1A1
SCHEMBL7753345 0.80 USP14 (0.52) SIGMAR1ALDH1A1USP14GAA
SCHEMBL8407956 0.80 ITGB3 (0.44) HRH3ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed