SCHEMBL8560217

SCHEMBL8560217

N=C(N)NS(=O)(=O)c1cnccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.41
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
CSNK1G2 P78368 1/20 0.41
CSNK1G1 Q9HCP0 1/20 0.41
LMNA P02545 2/20 0.39
CA12 O43570 6/20 0.38
CA2 P00918 6/20 0.38
CA9 Q16790 6/20 0.38
CA14 Q9ULX7 5/20 0.38
CA1 P00915 5/20 0.38
ALDH1A1 P00352 4/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9264558 0.85 BRS3 (0.39) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1
SCHEMBL1268486 0.77 POLB (0.51) CA12CA2CA9CA1ALDH1A1
SCHEMBL8555843 0.75 CA1 (0.32) CA12CA2CA9CA14CA1
SCHEMBL8212413 0.75 LMNA (0.49) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1
SCHEMBL8323021 0.72 ALDH1A1 (0.47) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1
SCHEMBL2879049 0.72 NAPRT (0.44) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1
SCHEMBL51312 0.72 CA12 (0.58) LMNACA12CA2CA9CA14
SCHEMBL13971307 0.71 CSNK1A1 (0.46) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1
SCHEMBL8560220 0.71 F2 (0.47) LMNACA12CA2CA9CA14
SCHEMBL7908992 0.71 GSTO1 (0.45) CSNK1A1CSNK1DCSNK1ECSNK1G2CSNK1G1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
US-5459138-A Dysfunctions of glutamatergic neurotransmission associated with learning and memory ADIR ET COMPAGNIE (FR) 1995-10-17 US disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed