SCHEMBL8560347

SCHEMBL8560347

CCOc1cc2c(Nc3ccc(Oc4ccccc4)cc3)ccnc2nc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.52
RAB9A P51151 2/20 0.42
FGFR2 P21802 2/20 0.42
POLB P06746 3/20 0.41
MAPT P10636 2/20 0.41
RAD52 P43351 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
RIPK2 O43353 1/20 0.41
EGFR P00533 1/20 0.41
EPHB2 P29323 1/20 0.41
SLC2A1 P11166 2/20 0.40
HTT P42858 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
EHMT2 Q96KQ7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8566240 0.99 ERBB2 (0.51) ERBB2RAB9AFGFR2POLBMAPT
SCHEMBL8325406 0.90 PDE10A (0.41) ERBB2RAB9AFGFR2POLBMAPT
Hydrochloric Acid SCHEMBL8468831 0.88 PDE10A (0.42) ERBB2RAB9AFGFR2POLBMAPT
SCHEMBL8559967 0.88 PDGFRA (0.48) RAB9AFGFR2POLBMAPTRAD52
Water SCHEMBL8328226 0.87 PDGFRA (0.47) RAB9AFGFR2POLBMAPTRAD52
Hydrochloric Acid SCHEMBL8566059 0.87 HTT (0.50) RAB9AFGFR2POLBMAPTRAD52
SCHEMBL9541717 0.86 MAPT (0.50) MAPTKDM4ETP53SMN1; SMN2THRB
SCHEMBL8567323 0.84 MAPKAPK2 (0.46) RAB9APOLBMAPTKMT2ANPSR1
SCHEMBL8327641 0.82 POLB (0.37) POLBKMT2AL3MBTL1RIPK2EGFR
SCHEMBL8568868 0.81 HRH3 (0.49) EHMT2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
EP-0618916-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES Knoll AG (DE) 1994-10-12 EP disclosed