SCHEMBL8567323

SCHEMBL8567323

CCOc1cc2c(Nc3ccc(O)cc3)ccnc2nc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 2/20 0.46
GAA P10253 3/20 0.43
MAPT P10636 2/20 0.43
ATM Q13315 2/20 0.43
EGFR P00533 4/20 0.38
POLB P06746 2/20 0.38
PTK6 Q13882 1/20 0.38
PDGFRA P16234 1/20 0.37
THRB P10828 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
KMT2A Q03164 1/20 0.37
PLEC Q15149 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
KDR P35968 2/20 0.37
GAK O14976 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324401 0.87 POLB (0.37) MAPKAPK2GAAMAPTEGFRPOLB
SCHEMBL8559967 0.87 PDGFRA (0.48) MAPTEGFRPOLBPTK6PDGFRA
SCHEMBL8561272 0.87 GAK (0.37) MAPKAPK2GAAMAPTEGFRPOLB
Hydrochloric Acid SCHEMBL8326683 0.86 POLB (0.36) MAPKAPK2GAAMAPTEGFRPOLB
Hydrochloric Acid SCHEMBL8566059 0.86 HTT (0.50) MAPTEGFRPOLBPTK6PDGFRA
Water SCHEMBL8328226 0.86 PDGFRA (0.47) MAPTEGFRPOLBPTK6PDGFRA
Hydrochloric Acid SCHEMBL8560744 0.86 GAK (0.36) MAPKAPK2GAAMAPTEGFRPOLB
SCHEMBL8327641 0.86 POLB (0.37) MAPKAPK2EGFRPOLBPTK6PDGFRA
SCHEMBL8566892 0.85 POLB (0.39) GAAMAPTATMEGFRPOLB
SCHEMBL8560347 0.84 ERBB2 (0.52) MAPKAPK2GAAMAPTEGFRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
WO-1993013097-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed