SCHEMBL8568868

SCHEMBL8568868

CCOc1cc2c(Nc3ccc(OCCN(CC)CC)cc3)ccnc2nc1C

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.49
ESR1 P03372 1/20 0.42
KDR P35968 1/20 0.42
SRC P12931 4/20 0.41
CDK4 P11802 2/20 0.39
CCND1 P24385 2/20 0.39
CCND2 P30279 2/20 0.39
CCND3 P30281 2/20 0.39
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39
WEE1 P30291 2/20 0.39
LCK P06239 2/20 0.38
EHMT2 Q96KQ7 1/20 0.38
BTK Q06187 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8561027 0.98 HRH3 (0.48) HRH3ESR1KDRSRCCDK4
SCHEMBL9540620 0.93 HRH3 (0.46) HRH3ESR1KDRSRCABL1
SCHEMBL8559967 0.84 PDGFRA (0.48) SRCABL1LCKEHMT2
Water SCHEMBL8328226 0.83 PDGFRA (0.47) LCKEHMT2
Hydrochloric Acid SCHEMBL8566059 0.83 HTT (0.50) LCKEHMT2
SCHEMBL8560347 0.81 ERBB2 (0.52) KDREHMT2
SCHEMBL8567323 0.81 MAPKAPK2 (0.46) KDRCDK4LCKEHMT2
Hydrochloric Acid SCHEMBL8566240 0.81 ERBB2 (0.51) KDREHMT2
SCHEMBL8565911 0.79 CDK4 (0.39) KDRCDK4ABL1LCKEHMT2
SCHEMBL8327641 0.79 POLB (0.37) SRCABL1LCKEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
EP-0618916-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES Knoll AG (DE) 1994-10-12 EP disclosed