SCHEMBL8560409

SCHEMBL8560409

O=C(Nc1ccc(C(=O)N2CCc3ccccc3-c3ccccc32)cc1)c1ccccc1OC(F)(F)F

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.53
AVPR1A P37288 3/20 0.53
OXTR P30559 2/20 0.53
NAMPT P43490 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558289 0.87 AVPR2 (0.60) AVPR2AVPR1AOXTR
SCHEMBL8560388 0.84 AVPR1A (0.60) AVPR2AVPR1AOXTRNAMPT
SCHEMBL8562670 0.82 AVPR1A (0.60) AVPR2AVPR1AOXTR
SCHEMBL8556989 0.82 AVPR1A (0.72) AVPR2AVPR1AOXTR
SCHEMBL8316224 0.81 AVPR2 (0.44) AVPR2AVPR1AOXTR
SCHEMBL8558555 0.81 AVPR2 (0.55) AVPR2AVPR1A
SCHEMBL8562680 0.81 ALDH1A1 (0.59) AVPR2AVPR1AOXTRNAMPT
SCHEMBL8557460 0.81 AVPR1A (0.64) AVPR2AVPR1AOXTR
SCHEMBL8557218 0.80 AVPR1A (0.60) AVPR2AVPR1AOXTRNAMPT
SCHEMBL8559797 0.80 RAB9A (0.55) AVPR2AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed