SCHEMBL8560521

SCHEMBL8560521

C=CCc1c(C)c(C)c2c(c1O)C(C)(C)C(=O)N2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
NPSR1 Q6W5P4 1/20 0.34
HPGD P15428 2/20 0.32
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560875 0.74 MEN1 (0.36) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL8556883 0.71 PDK2 (0.40) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL20088306 0.67 IMPDH2 (0.34) ALDH1A1NPSR1HPGDKDM4EGLA
SCHEMBL8554202 0.67 MEN1 (0.35) ALDH1A1HPGDKDM4EGAA
SCHEMBL8598630 0.66 MEN1 (0.34) HPGDKDM4EGAA
SCHEMBL8555558 0.65 GABRA1 (0.42) NPSR1HPGDKDM4EGAAL3MBTL1
SCHEMBL5810793 0.63 KDM4E (0.39) ALDH1A1NPSR1HPGDKDM4EGLA
SCHEMBL8555174 0.62 PDK2 (0.31)
SCHEMBL8556416 0.62
SCHEMBL8557831 0.62 ALDH1A1 (0.36) ALDH1A1HPGDKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
US-5510366-A INOTROPIC, ANTIARRHYMTHMIA AGENTS, VASODILATORS KOWA CO., LTD. (JP) 1996-04-23 US disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed