SCHEMBL8561322

SCHEMBL8561322

CC(C)(C)OC(=O)N[C@@]1(OC(=O)OCc2ccccc2)CCc2cccc(O)c2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.40
GHSR Q92847 1/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 1/20 0.37
ACHE P22303 1/20 0.37
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CTSL P07711 1/20 0.35
PPARA Q07869 1/20 0.34
HTR1A P08908 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
CA12 O43570 1/20 0.33
CA7 P43166 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KLK7 P49862 1/20 0.33
KLK5 Q9Y337 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569271 0.87 GHSR (0.39) GHSRCA1CA2ACHEHTR1A
SCHEMBL8520181 0.87 CA1 (0.41) CA1CA2ACHECTSLCA12
SCHEMBL8560312 0.86 GHSR (0.39) GHSRCA1CA2ACHEHTR1A
SCHEMBL8559137 0.86 GHSR (0.39) GHSRCA1CA2ACHEHTR1A
SCHEMBL8997648 0.86 SYK (0.38) SYKGHSRCA1CA2ACHE
SCHEMBL8569372 0.85 GHSR (0.39) GHSRCA1CA2ACHEHTR1A
SCHEMBL8576152 0.85 GHSR (0.39) GHSRCA1CA2ACHEHTR1A
SCHEMBL8997699 0.83 CA1 (0.36) SYKGHSRCA1CA2ACHE
SCHEMBL8575729 0.82 CA1 (0.39) SYKGHSRCA1CA2ACHE
SCHEMBL8567143 0.82 CA1 (0.39) SYKGHSRCA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640618-B1 Tetrahydronaphthalene-peptide derivatives HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed
EP-0640618-A1 Tetrahydronaphthalene-peptide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-03-01 EP disclosed