SCHEMBL8520181

SCHEMBL8520181

COC(=O)O[C@@]1(NC(=O)OCc2ccccc2)CCc2cccc(O)c2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
ACHE P22303 1/20 0.41
CYP3A4 P08684 7/20 0.39
TSHR P16473 6/20 0.39
CYP2C9 P11712 6/20 0.39
CYP2C19 P33261 5/20 0.39
ALDH1A1 P00352 4/20 0.39
CYP1A2 P05177 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CASP1 P29466 1/20 0.38
KYNU Q16719 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561322 0.87 SYK (0.40) CA1CA2ACHECTSLCA12
SCHEMBL8560312 0.81 GHSR (0.39) CA1CA2ACHE
SCHEMBL8559137 0.81 GHSR (0.39) CA1CA2ACHE
SCHEMBL8583599 0.80 CTSS (0.44) CA1CA2ACHECTSLCTSB
SCHEMBL8426423 0.80 CTSS (0.44) CA1CA2ACHECTSLCTSB
SCHEMBL8567143 0.78 CA1 (0.39) CA1CA2ACHECYP3A4TSHR
SCHEMBL8575729 0.78 CA1 (0.39) CA1CA2ACHECYP3A4TSHR
SCHEMBL8997600 0.77 SYK (0.40) CA1CA2ACHECYP3A4CYP2C9
SCHEMBL8569271 0.76 GHSR (0.39) CA1CA2ACHE
SCHEMBL8569372 0.74 GHSR (0.39) CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640618-B1 Tetrahydronaphthalene-peptide derivatives HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed
EP-0640618-A1 Tetrahydronaphthalene-peptide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-03-01 EP disclosed