SCHEMBL8561372

SCHEMBL8561372

CN(CC(OCCOS(C)(=O)=O)c1ccc(Cl)c(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F2R P25116 2/20 0.34
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 3/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
FFAR1 O14842 1/20 0.31
TACR2 P21452 2/20 0.31
S1PR3 Q99500 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KAT6A Q92794 1/20 0.31
KAT5 Q92993 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557969 0.86 SLC6A2 (0.37) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL8970527 0.84 F2R (0.34) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL7306571 0.83 TACR2 (0.40) TACR2
SCHEMBL8563201 0.78 SLC6A3 (0.43) SLC6A2SLC6A4SLC6A3TACR2LMNA
SCHEMBL8559300 0.77 F2R (0.52) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL8565799 0.75 TACR1 (0.40) CYP3A4CYP2D6FFAR1
SCHEMBL8970508 0.74 TACR2 (0.57) TACR2
SCHEMBL8483223 0.74 TACR2 (0.41) F2RTACR2
SCHEMBL4870085 0.73 TACR2 (0.46) TACR2
SCHEMBL756561 0.73 TACR2 (0.46) TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726313-A Substituted arylaliphatic compounds, method of preparing them and pharmaceutical compositions in which they are present SANOFI (FR) 1998-03-10 US disclosed
EP-0700386-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1996-03-13 EP disclosed
WO-1995026338-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1995-10-05 WO disclosed