SCHEMBL8557969

SCHEMBL8557969

CN(CC(OCCO)c1ccc(Cl)c(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
F2R P25116 1/20 0.36
TACR2 P21452 5/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FFAR1 O14842 1/20 0.34
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561372 0.86 F2R (0.34) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL4870085 0.81 TACR2 (0.46) TACR2
SCHEMBL756561 0.81 TACR2 (0.46) TACR2
SCHEMBL8559300 0.81 F2R (0.52) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8563201 0.81 SLC6A3 (0.43) SLC6A2SLC6A4SLC6A3TACR2LMNA
SCHEMBL8970883 0.80 F2R (0.36) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL7315171 0.80 TACR2 (0.45) TACR2
SCHEMBL8970508 0.78 TACR2 (0.57) TACR2
SCHEMBL8483223 0.78 TACR2 (0.41) F2RTACR2
SCHEMBL4865304 0.76 TACR2 (0.39) F2RTACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726313-A Substituted arylaliphatic compounds, method of preparing them and pharmaceutical compositions in which they are present SANOFI (FR) 1998-03-10 US disclosed
EP-0700386-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1996-03-13 EP disclosed
WO-1995026338-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1995-10-05 WO disclosed