SCHEMBL8561776

SCHEMBL8561776

COc1ccc(C(=O)N(C)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
TSHR P16473 4/20 0.44
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559862 0.90 AVPR2 (0.45) SMN1; SMN2RAB9AALDH1A1MAPTTUBB4A
SCHEMBL8557707 0.89 ALDH1A1 (0.47) SMN1; SMN2RAB9ATSHRALDH1A1TUBB4A
SCHEMBL7337838 0.85 AVPR1A (0.58) AVPR2AVPR1A
SCHEMBL8558249 0.82 NPC1 (0.45) SMN1; SMN2RAB9AKMT2AHSP90AA1PDK1
SCHEMBL8558262 0.80 AVPR1A (0.40) SMN1; SMN2RAB9AALDH1A1KMT2AHSP90AA1
SCHEMBL8561629 0.80 AVPR2 (0.52) SMN1; SMN2RAB9AKMT2AAVPR2AVPR1A
SCHEMBL8561048 0.80 AVPR2 (0.48) HSP90AA1PDK1AVPR2AVPR1A
SCHEMBL8562797 0.80 AVPR2 (0.54) HSP90AA1PDK1AVPR2AVPR1A
SCHEMBL8559548 0.79 POLB (0.51) ALDH1A1LMNAHSP90AA1PDK1AVPR2
SCHEMBL8561685 0.79 AVPR1A (0.44) SMN1; SMN2RAB9AKMT2AHSP90AA1PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed