SCHEMBL8561859

SCHEMBL8561859

CC(C)(C)OC(=O)c1ccc(CN2CCC(Br)C2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.49
SIRT1 Q96EB6 1/20 0.49
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
TP53 P04637 1/20 0.42
KDM1A O60341 5/20 0.42
SRC P12931 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ROCK2 O75116 1/20 0.39
CHKA P35790 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
THRB P10828 1/20 0.38
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25023516 0.84 SIRT2 (0.48) SIRT2SIRT1HDAC1HDAC6TP53
SCHEMBL8569448 0.82 DRD2 (0.45) TP53KDM4EHDAC8THRB
SCHEMBL27485081 0.80 PTGS1 (0.46) HDAC1HDAC6KDM1AKDM4EHDAC8
Bromide SCHEMBL8565335 0.78 SIRT2 (0.48) SIRT2SIRT1HDAC1HDAC6TP53
SCHEMBL8563968 0.78 HDAC8 (0.40) HDAC1HDAC6TP53HDAC8
SCHEMBL8563972 0.78 TP53 (0.37) HDAC1HDAC6TP53ROCK2ELANE
SCHEMBL3689873 0.78 HRH3 (0.55) HDAC1HDAC6KDM4ECHKAHDAC8
SCHEMBL28176279 0.78 HRH3 (0.55) HDAC1HDAC6KDM4ECHKAHDAC8
SCHEMBL15033023 0.76 KDM4E (0.50) SIRT2SIRT1HDAC1HDAC6KDM1A
SCHEMBL28175300 0.76 KDM4E (0.50) SIRT2SIRT1HDAC1HDAC6KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed