SCHEMBL8563972

SCHEMBL8563972

CC(C)(C)OC(CCC(=O)O)=Nc1ccc(CN2CCC(Br)C2=O)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.37
ROCK2 O75116 1/20 0.35
NPFFR1 Q9GZQ6 2/20 0.34
NPFFR2 Q9Y5X5 2/20 0.34
KCNH2 Q12809 1/20 0.33
ELANE P08246 1/20 0.33
LMNA P02545 1/20 0.33
VEGFA P15692 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561859 0.78 SIRT2 (0.49) TP53ROCK2ELANEHDAC1HDAC6
SCHEMBL8569448 0.75 DRD2 (0.45) TP53
SCHEMBL8563968 0.73 HDAC8 (0.40) TP53HDAC1HDAC6
SCHEMBL27485081 0.71 PTGS1 (0.46) HDAC1HDAC6
SCHEMBL16874550 0.69 KCNH2 (0.51) TP53KCNH2LMNA
SCHEMBL8564264 0.69 DDB1 (0.50) HDAC1HDAC6
SCHEMBL8564268 0.69 DDB1 (0.50) HDAC1HDAC6
SCHEMBL8560205 0.69 KDM4E (0.54) KCNH2HDAC1
SCHEMBL8562132 0.69 GAA (0.56) LMNA
SCHEMBL8560210 0.69 KDM4E (0.54) KCNH2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed