SCHEMBL8569448

SCHEMBL8569448

CC(C)(C)OC(=O)Nc1ccc(CN2CCC(Br)C2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.45
CYP17A1 P05093 1/20 0.45
HDAC3 O15379 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
FPR2 P25090 1/20 0.42
PRKDC P78527 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK14 Q16539 1/20 0.41
NPY1R P25929 1/20 0.41
NAMPT P43490 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TNIK Q9UKE5 1/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563968 0.86 HDAC8 (0.40) HDAC3HDAC8NCOR2FPR2ALDH1A1
SCHEMBL8561859 0.82 SIRT2 (0.49) HDAC8KDM4ETP53THRB
SCHEMBL27520459 0.82 TNIK (0.46) HDAC8FPR2KDM4EALDH1A1TNIK
SCHEMBL28802622 0.80 KDM4E (0.63) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL7597673 0.80 ROCK2 (0.56) DRD2CYP17A1FPR2PRKDCNAMPT
SCHEMBL1604864 0.79 KDM4E (0.66) DRD2CYP17A1KDM4EALDH1A1KMT2A
SCHEMBL8563972 0.75 TP53 (0.37) TP53
SCHEMBL6583535 0.75 BCHE (0.52) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL7375302 0.75 DRD2 (0.52) DRD2PTGDR2CYP17A1HDAC3HDAC8
SCHEMBL22571323 0.75 CD274 (0.61) ALDH1A1MEN1KMT2ACD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed