SCHEMBL7418940

SCHEMBL7418940

O=C1CCC(n2ccn(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)c2=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.42
ESR2 Q92731 8/20 0.42
HDAC6 Q9UBN7 1/20 0.33
PKM P14618 1/20 0.33
ABHD6 Q9BV23 3/20 0.31
TYRO3 Q06418 1/20 0.31
MERTK Q12866 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415517 0.84 DRD2 (0.43)
SCHEMBL8562237 0.83 ESR1 (0.39) ESR1ESR2HDAC6ABHD6
SCHEMBL8562233 0.83 ESR1 (0.39) ESR1ESR2HDAC6ABHD6
SCHEMBL8564898 0.82 ESR1 (0.39) ESR1ESR2HDAC6ABHD6
SCHEMBL8564893 0.82 ESR1 (0.39) ESR1ESR2HDAC6ABHD6
SCHEMBL7472118 0.72 ESR1 (0.41) ESR1ESR2HDAC6
SCHEMBL7472374 0.71 TMEM97 (0.43) ESR1ESR2
SCHEMBL7476930 0.69 DRD2 (0.32)
SCHEMBL7476926 0.69 DRD2 (0.32)
SCHEMBL8562345 0.69 ESR1 (0.39) ESR1ESR2HDAC6ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed