SCHEMBL8558246

SCHEMBL8558246

O=C(Nc1ccc(C(=O)N2c3ccccc3CNc3ccccc32)c(Cl)c1)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.48
AVPR1A P37288 7/20 0.48
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
RORC P51449 2/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TYK2 P29597 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
EPHX2 P34913 1/20 0.38
OXTR P30559 1/20 0.38
IL2 P60568 1/20 0.37
NPY2R P49146 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562699 0.90 AVPR2 (0.39) AVPR2AVPR1AITGB1ITGA4RORC
SCHEMBL8564681 0.88 AVPR2 (0.42) AVPR2AVPR1ATYK2HPGD
SCHEMBL8562616 0.86 ITGB1 (0.40) AVPR2AVPR1AITGB1ITGA4RORC
SCHEMBL8561799 0.84 AVPR2 (0.59) AVPR2AVPR1ANPC1RAB9ASMN1; SMN2
SCHEMBL8561421 0.83 AVPR2 (0.56) AVPR2AVPR1AOXTR
SCHEMBL8559867 0.81 RAB9A (0.47) AVPR2AVPR1ARAB9A
SCHEMBL8556908 0.81 RAB9A (0.47) AVPR2AVPR1ANPC1RAB9A
SCHEMBL8561432 0.81 AVPR2 (0.55) AVPR2AVPR1ANPC1RAB9ATYK2
SCHEMBL8562470 0.80 AVPR2 (0.40) AVPR2AVPR1ATYK2
SCHEMBL8557787 0.80 PNLIP (0.50) AVPR2AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed