SCHEMBL8563173

SCHEMBL8563173

Nc1nc(NCC2CC2)c2[nH]cnc2n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 5/20 0.58
NUDT1 P36639 1/20 0.55
PRKACA P17612 3/20 0.54
CDK2 P24941 5/20 0.51
CCNB1 P14635 4/20 0.51
CCNA2 P20248 4/20 0.51
CCNA1 P78396 4/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
CCNB2 O95067 1/20 0.50
MAPK3 P27361 1/20 0.50
CLK1 P49759 1/20 0.50
CDK5 Q00535 1/20 0.50
PIN1 Q13526 1/20 0.50
CCNB3 Q8WWL7 1/20 0.50
MAP3K5 Q99683 1/20 0.50
PDPK1 O15530 1/20 0.49
GDA Q9Y2T3 1/20 0.49
CHUK O15111 1/20 0.48
BRAF P15056 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16147021 0.79 CDK1 (0.63) CDK1NUDT1PRKACACDK2CCNB1
SCHEMBL8563169 0.78 CHUK (0.52) CDK1PRKACACDK2CCNB1CCNA2
SCHEMBL9205057 0.78 HTT (0.59) CDK2
SCHEMBL10838746 0.78 NUDT1 (0.67) CDK1NUDT1PRKACACDK2HDAC1
SCHEMBL133157 0.78 LMNA (0.54) CDK1NUDT1CDK2PDPK1GDA
SCHEMBL16146456 0.77 NUDT1 (0.65) CDK1NUDT1PRKACACDK2CCNB1
SCHEMBL7626878 0.75 LMNA (0.58) CDK1CDK2CCNB1CCNA2CCNA1
SCHEMBL796828 0.75 CDK1 (0.59) CDK1NUDT1PRKACACDK2CCNB1
SCHEMBL7621600 0.75 LMNA (0.62) CDK1CDK2CCNB1CCNA2CCNA1
SCHEMBL16146485 0.75 CDK1 (0.59) CDK1NUDT1PRKACACDK2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817639-A VIRICIDES YAMASA CORPORATION (JP) 1998-10-06 US disclosed
US-5811408-A ANTITUMOR AND ANTICARCINOGENIC AGENT; INTRODUCING SULFONYL GROUP ON HYDROXY GROUP OF TETRAHYDROFURAN RING, HYDROLYSIS, BLOCKING, OXIDATION, WITTING REACTION, DEPROTECTION AND PHOSPHORYLATION YAMASA CORPORATION (JP) 1998-09-22 US disclosed
EP-0770621-A1 2'-DEOXY-2'-(SUBSTITUTED OR UNSUBSTITUTED METHYLIDENE)-4'-THIONUCLEOSIDE YAMASA CORPORATION (JP) 1997-05-02 EP disclosed