SCHEMBL8563180

SCHEMBL8563180

Nc1nc(N)c2c(n1)CCC2CCCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 9/20 0.51
GART P22102 9/20 0.51
ATIC P31939 4/20 0.50
FOLR2 P14207 3/20 0.50
SLC46A1 Q96NT5 6/20 0.49
SLC19A1 P41440 4/20 0.49
SHMT1 P34896 2/20 0.48
SHMT2 P34897 2/20 0.48
DHFR P00374 1/20 0.47
MTR Q99707 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001769 0.93 FOLR1 (0.49) FOLR1GARTATICFOLR2SLC46A1
SCHEMBL9001752 0.87 GART (0.53) FOLR1GARTATICFOLR2SLC46A1
SCHEMBL9439570 0.86 GART (0.58) FOLR1GARTATICFOLR2SLC46A1
SCHEMBL1066004 0.85 DHFR (0.59) GARTATICDHFRMTR
SCHEMBL8565987 0.84 FOLR2 (0.49) FOLR1ATICFOLR2DHFRMTR
SCHEMBL8566521 0.84 DHFR (0.46) GARTDHFRMTR
SCHEMBL8566814 0.83 FOLR1 (0.39) FOLR1DHFRMTR
SCHEMBL8567075 0.82 DHFR (0.47) GARTDHFRMTR
SCHEMBL8571475 0.81 DHFR (0.57) GARTDHFRMTR
SCHEMBL8568731 0.81 DHFR (0.47) FOLR1ATICFOLR2DHFRMTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed