SCHEMBL8565987

SCHEMBL8565987

Nc1nc(N)c2c(n1)CCC2CCCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)o1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FOLR2 P14207 1/20 0.49
FOLR1 P15328 1/20 0.49
ATIC P31939 1/20 0.49
DHFR P00374 9/20 0.46
MTR Q99707 1/20 0.46
TYMS P04818 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568731 0.95 DHFR (0.47) FOLR2FOLR1ATICDHFRMTR
SCHEMBL9001930 0.93 ATIC (0.48) FOLR2FOLR1ATICDHFRMTR
SCHEMBL9001791 0.88 ATIC (0.46) FOLR2FOLR1ATICDHFRMTR
SCHEMBL1066004 0.87 DHFR (0.59) ATICDHFRMTR
SCHEMBL8563180 0.84 FOLR1 (0.51) FOLR2FOLR1ATICDHFRMTR
SCHEMBL8571475 0.84 DHFR (0.57) DHFRMTR
SCHEMBL9001799 0.80 DHFR (0.54) ATICDHFRMTRTYMS
SCHEMBL8571393 0.77 ATIC (0.59) ATICDHFRMTR
SCHEMBL9001769 0.77 FOLR1 (0.49) FOLR2FOLR1ATIC
SCHEMBL8603963 0.77 DHFR (0.55) DHFRMTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed