SCHEMBL8563606

SCHEMBL8563606

COC(=O)[C@H](Cc1cc(OC)cc(OC)c1)NC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 2/20 0.48
POLB P06746 2/20 0.47
TACR1 P25103 2/20 0.46
MTNR1A P48039 3/20 0.43
MTNR1B P49286 3/20 0.43
ATM Q13315 1/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
APEX1 P27695 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
LCK P06239 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563604 1.00 KMT2A (0.49) KMT2AALDH1A1POLBTACR1MTNR1A
SCHEMBL8567267 0.88 ITGB3 (0.50) KMT2AALDH1A1POLBMTNR1AMTNR1B
SCHEMBL8567271 0.88 ITGB3 (0.50) KMT2AALDH1A1POLBMTNR1AMTNR1B
SCHEMBL6139248 0.85 POLB (0.61) KMT2AALDH1A1POLBTACR1MTNR1A
SCHEMBL30082808 0.85 POLB (0.61) KMT2AALDH1A1POLBTACR1MTNR1A
SCHEMBL5706152 0.84 ACACB (0.58) KMT2AALDH1A1TACR1ATMHSD17B10
SCHEMBL6662892 0.84 ACACB (0.58) KMT2AALDH1A1TACR1ATMHSD17B10
SCHEMBL10477398 0.82 CYP3A4 (0.42) KMT2APOLBTACR1MTNR1AMTNR1B
SCHEMBL2674354 0.82 ALDH1A1 (0.49) KMT2AALDH1A1TACR1MEN1
SCHEMBL2674352 0.82 ALDH1A1 (0.49) KMT2AALDH1A1TACR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed
US-4058642-A HYPERTENSIVE BOEHRINGER INGELHEIM GMBH (DT) 1977-11-15 US disclosed