SCHEMBL8563690

SCHEMBL8563690

COc1cccc(N2CCC(Br)C2=O)c1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.48
MAPT P10636 1/20 0.48
MCHR1 Q99705 2/20 0.42
KMT2A Q03164 1/20 0.41
GRM2 Q14416 1/20 0.40
POLB P06746 1/20 0.40
KCNH2 Q12809 2/20 0.40
OPRM1 P35372 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
CTSG P08311 1/20 0.39
CMA1 P23946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568619 0.90 ROCK2 (0.56) ROCK2MAPTMCHR1KMT2AKCNH2
SCHEMBL8568624 0.90 ROCK2 (0.56) ROCK2MAPTMCHR1KMT2AKCNH2
SCHEMBL1514921 0.76 MEN1 (0.50) ROCK2KMT2APOLBSIGMAR1
SCHEMBL8285848 0.74 ROCK2 (0.53) ROCK2MAPTMCHR1KMT2AGRM2
SCHEMBL14301512 0.74 ROCK2 (0.53) ROCK2MAPTMCHR1KMT2AKCNH2
SCHEMBL8788607 0.74 DRD2 (0.50) ROCK2MCHR1KCNH2DRD2DRD3
SCHEMBL892458 0.74 ROCK2 (0.53) ROCK2MAPTMCHR1KMT2APOLB
SCHEMBL892517 0.74 ROCK2 (0.53) ROCK2MAPTMCHR1KMT2APOLB
Bromide SCHEMBL8897811 0.72 MAPT (0.49) ROCK2MAPTMCHR1KMT2AGRM2
Bromide SCHEMBL8563694 0.72 MAPT (0.49) ROCK2MAPTMCHR1KMT2AGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed