SCHEMBL8568624

SCHEMBL8568624

COc1cccc(N2CC[C@H](Br)C2=O)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.56
MAPT P10636 2/20 0.50
KMT2A Q03164 1/20 0.48
MCHR1 Q99705 1/20 0.47
MGLL Q99685 1/20 0.46
DRD2 P14416 2/20 0.45
DRD3 P35462 2/20 0.45
ALOX5 P09917 1/20 0.45
KCNH2 Q12809 1/20 0.45
FADS1 O60427 1/20 0.44
ADRB1 P08588 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568619 1.00 ROCK2 (0.56) ROCK2MAPTKMT2AMCHR1MGLL
SCHEMBL8563690 0.90 ROCK2 (0.48) ROCK2MAPTKMT2AMCHR1DRD2
SCHEMBL14301512 0.82 ROCK2 (0.53) ROCK2MAPTKMT2AMCHR1MGLL
SCHEMBL8285848 0.82 ROCK2 (0.53) ROCK2MAPTKMT2AMCHR1MGLL
SCHEMBL8788607 0.82 DRD2 (0.50) ROCK2MCHR1DRD2DRD3KCNH2
SCHEMBL28758908 0.80 GAA (0.55) MAPTKMT2AGAA
SCHEMBL892517 0.79 ROCK2 (0.53) ROCK2MAPTKMT2AMCHR1MGLL
SCHEMBL892458 0.79 ROCK2 (0.53) ROCK2MAPTKMT2AMCHR1MGLL
SCHEMBL8560581 0.79 FADS1 (0.45) ROCK2MAPTKMT2AMGLLDRD2
SCHEMBL8560582 0.79 FADS1 (0.45) ROCK2MAPTKMT2AMGLLDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed