SCHEMBL8563723

SCHEMBL8563723

Clc1ccn2c1cnc1c(N3CCSCC3)cccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.39
LCK P06239 1/20 0.34
POLB P06746 1/20 0.34
DRD3 P35462 4/20 0.33
DRD4 P21917 2/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
ALDH1A1 P00352 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK10 P53779 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DRD2 P14416 3/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRB1 P08588 1/20 0.31
LGMN Q99538 1/20 0.31
PRKDC P78527 1/20 0.30
KMT2A Q03164 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562733 0.84 DRD2 (0.49) DRD3DRD4HSD17B10DRD2HTR2A
SCHEMBL8562645 0.84 DRD2 (0.49) DRD3DRD4DRD2HTR2AHTR2C
SCHEMBL8565094 0.83 DHFR (0.40) LCKPOLBDRD3DRD4ALDH1A1
SCHEMBL8571229 0.80 ALDH1A1 (0.44) CNR2POLBALDH1A1ALOX15MAPK10
SCHEMBL8563995 0.79 DRD2 (0.54) DRD3DRD4DRD2HTR2AHTR2C
SCHEMBL8569163 0.79 GRM2 (0.45)
SCHEMBL8566284 0.79 DRD4 (0.54) DRD3DRD4ALDH1A1DRD2HTR2C
SCHEMBL8570952 0.78 HTR1A (0.43) DRD3DRD4MAPK10DRD2HTR2A
SCHEMBL8571687 0.77 HTR1A (0.49) DRD3DRD4DRD2HTR2C
SCHEMBL8880284 0.76 DHFR (0.50) POLBALDH1A1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed