SCHEMBL8563850

SCHEMBL8563850

CCCCCC(=O)NC(Cc1ccc(N2CCN(c3ccc4c(c3)CCNCC4)C2=O)cc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.52
ITGA2B P08514 8/20 0.52
FAAH O00519 2/20 0.45
ALDH1A1 P00352 1/20 0.42
ACE P12821 3/20 0.41
ACE2 Q9BYF1 3/20 0.41
S1PR1 P21453 1/20 0.39
GNAI3 P08754 1/20 0.38
GNAO1 P09471 1/20 0.38
GNAI1 P63096 1/20 0.38
PSMB5 P28074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8558942 0.82 S1PR1 (0.41) ITGB3ITGA2BS1PR1
Hydrochloric Acid SCHEMBL7396964 0.79 ITGB3 (0.51) ITGB3ITGA2BFAAHALDH1A1S1PR1
Hydrochloric Acid SCHEMBL8562284 0.79 HTR6 (0.40) S1PR1
SCHEMBL8565331 0.78 ITGB3 (0.40) ITGB3ITGA2BFAAHACEACE2
SCHEMBL8562408 0.77 S1PR1 (0.44) ITGB3ITGA2BS1PR1
Hydrochloric Acid SCHEMBL8564109 0.74 S1PR1 (0.47) S1PR1
Hydrochloric Acid SCHEMBL8564486 0.74 HTR6 (0.44) ITGB3ITGA2BS1PR1
SCHEMBL8559578 0.73 HTR6 (0.42) S1PR1
Hydrochloric Acid SCHEMBL8566255 0.73 HTR6 (0.41) S1PR1
SCHEMBL8565326 0.72 ITGB3 (0.40) ITGB3ITGA2BFAAHALDH1A1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed